About Drug Discovery Chemistry

Today’s Synthetic Molecules for Tomorrow’s Therapeutics

April 19-21, 2027 | Hilton San Diego Bayfront | San Diego, CA + Virtual

Focused on the discovery and optimization challenges of small-molecule and macrocyclic drug candidates, the 27th Annual Drug Discovery Chemistry explores the critical "middle space" of drug discovery—from hit identification and lead optimization to emerging modalities, AI-enabled design, and translational strategies. Join a community of discovery scientists and share the innovations shaping the next generation of medicines.

What is Drug Discovery Chemistry Europe?

A curated in-person and virtual conference for drug discovery scientists seeking practical insights and cross-disciplinary collaboration. The program is structured around themes including AI/ML, Degraders and Molecular Glues, Emerging Technology, Targeting PPI Interactions, DNA-Encoded Libraries, and new this year – Linker & Conjugation Chemistries.

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The Drug Discovery Chemistry Experience

The 2026 edition of Drug Discovery Chemistry Europe brought together scientists from across pharma, biotech, and academia, including Amgen, Roche, AstraZeneca, Novartis, Merck, GSK, and leading research institutions worldwide. View 2026 Attendees >>

Attendees consistently highlight the strong balance of high-quality science and networking, with one describing it as “the top conference for drug discovery... The most interesting tracks and talks in the field” and another noting “This event is the best for networking.” The meeting is designed to encourage interaction through poster sessions, networking breaks, and informal discussions that connect industry and academic perspectives.

Set in San Diego (also available virtually), the conference benefits from a vibrant scientific and cultural hub that enhances connection and collaboration throughout the event. Check out the venue >>