Drug Discovery Chemistry is now accepting speaker proposals for the premier event dedicated to medicinal, biophysical, and computational chemists working across pharma, biotech, and academia. Focused on the discovery and optimization challenges of small-molecule and macrocyclic drug candidates, the 27th Annual conference explores the critical "middle space" of drug discovery—from hit identification and lead optimization to emerging modalities, AI-enabled design, and translational strategies. Join a community of discovery scientists and share the innovations shaping the next generation of medicines.
Matthew Disney, PhDInstitute Professor & Chair,UF Scripps
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"Really the top conference for drug discovery in my view. The most interesting tracks and talks in the field."
Jörg S., ETH Zürich
"Drug Discovery Chemistry is a must attend event. It consistently has great speakers and attendees!"
Casey K., Professor, Purdue University
"The coverage of fascinating topics and the combination of industry and academic participants make this my favorite conference of the year!"
Christian H., École Polytechnique Fédérale de Lausanne
Based on highlights from our 2026 event
160
850
85+
100+
40+
25
DRUG DISCOVERY CHEMISTRY 2027
Returns to the Hilton San Diego Bayfront!
Hilton San Diego Bayfront
One Park Blvd.San Diego, CA 92101Phone: 619-564-3333
Conference Room Rate: $339 per night (single/double occupancy)
Hotel Reservation Deadline: March 22, 2027
We encourage attendees to book early, as rooms at the conference rate are available on a first-come, first-served basis through the reservation deadline.
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